Ident. | Authors (with country if any) | Title |
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002112 |
Clément Thomas [France] ; Johnny Vercouillie [France] ; Aurélie Doméné [France] ; Clovis Tauber [France] ; Michael Kassiou [Australie] ; Denis Guilloteau [France] ; Christophe Destrieux [France] ; Sophie Sérrière [France] ; Sylvie Chalon [France] | Detection of Neuroinflammation in a Rat Model of Subarachnoid Hemorrhage Using [18F]DPA-714 PET Imaging |
003185 |
Sophie Sérrière [France] ; Clovis Tauber [France] ; Johnny Vercouillie [France] ; Céline Mothes [France] ; Christelle Pruckner [France] ; Denis Guilloteau [France] ; Michael Kassiou [Australie] ; Aurélie Doméné [France] ; Lucette Garreau [France] ; Guylène Page [France] ; Sylvie Chalon [France] | Amyloid load and translocator protein 18 kDa in APPswePS1-dE9 mice: a longitudinal study. |
003A79 |
Maria-Joao Ribeiro [France] ; Johnny Vercouillie [France] ; Severine Debiais [France] ; Jean-Philippe Cottier [France] ; Isabelle Bonnaud [France] ; Vincent Camus [France] ; Samuel Banister [Australie] ; Michael Kassiou [Australie] ; Nicolas Arlicot [France] ; Denis Guilloteau [France] | Could 18 F-DPA-714 PET imaging be interesting to use in the early post-stroke period? |
003C80 |
Vincent Médran-Navarrete [France] ; Nicholas Bernards [France] ; Bertrand Kuhnast [France] ; Annelaure Damont [France] ; Géraldine Pottier [France] ; Marie-Anne Peyronneau [France] ; Michael Kassiou [Australie] ; Frank Marguet [France] ; Frédéric Puech [France] ; Raphaël Boisgard [France] ; Frédéric Dollé [France] | [18F]DPA‐C5yne, a novel fluorine‐18‐labelled analogue of DPA‐714: radiosynthesis and preliminary evaluation as a radiotracer for imaging neuroinflammation with PET |
004399 |
Hervé Boutin [Royaume-Uni] ; Christian Prenant [Royaume-Uni] ; Renaud Maroy [France] ; James Galea [Royaume-Uni] ; Andrew D. Greenhalgh [Royaume-Uni] ; Alison Smigova [Royaume-Uni] ; Christopher Cawthorne [Royaume-Uni] ; Peter Julyan [Royaume-Uni] ; Shane M. Wilkinson [Australie] ; Samuel D. Banister [Australie] ; Gavin Brown [Royaume-Uni] ; Karl Herholz [Royaume-Uni] ; Michael Kassiou [Australie] ; Nancy J. Rothwell [Royaume-Uni] | [18F]DPA-714: Direct Comparison with [11C]PK11195 in a Model of Cerebral Ischemia in Rats |
005B37 |
Nicolas Arlicot [France] ; Johnny Vercouillie [France] ; Maria-João Ribeiro [France] ; Clovis Tauber [France] ; Yann Venel [France] ; Jean-Louis Baulieu [France] ; Serge Maia [France] ; Philippe Corcia [France] ; Michael G. Stabin [États-Unis] ; Aaron Reynolds [Australie] ; Michael Kassiou [Australie] ; Denis Guilloteau [France] | Initial evaluation in healthy humans of [18F]DPA-714, a potential PET biomarker for neuroinflammation |
006216 |
Caroline Drake [Royaume-Uni] ; Hervé Boutin [Royaume-Uni] ; Matthew S. Jones [Royaume-Uni] ; Adam Denes [Royaume-Uni] ; Barry W. Mccoll [Royaume-Uni] ; Johann R. Selvarajah [Royaume-Uni] ; Sharon Hulme [Royaume-Uni] ; Rachel F. Georgiou [Royaume-Uni] ; Rainer Hinz [Royaume-Uni] ; Alexander Gerhard [Royaume-Uni] ; Andy Vail [Royaume-Uni] ; Christian Prenant [Royaume-Uni] ; Peter Julyan [Royaume-Uni] ; Renaud Maroy [France] ; Gavin Brown [Royaume-Uni] ; Alison Smigova [Royaume-Uni] ; Karl Herholz [Royaume-Uni] ; Michael Kassiou [Australie] ; David Crossman [Royaume-Uni] ; Sheila Francis [Royaume-Uni] ; Spencer D. Proctor [Canada] ; James C. Russell [Canada] ; Stephen J. Hopkins [Royaume-Uni] ; Pippa J. Tyrrell [Royaume-Uni] ; Nancy J. Rothwell [Royaume-Uni] ; Stuart M. Allan [Royaume-Uni] | Brain inflammation is induced by co-morbidities and risk factors for stroke |
006684 |
Annelaure Damont [France] ; Raphael Boisgard [France] ; Bertrand Kuhnast [France] ; Frederic Lemee [France] ; Guillaume Raggiri [France] ; Alana M. Scarf [Australie] ; Eleonora Da Pozzo [Italie] ; Silvia Selleri [Italie] ; Claudia Martini [Italie] ; Bertrand Tavitian [France] ; Michael Kassiou [Australie] ; Frederic Dolle [France] | Synthesis of 6-[18F]fluoro-PBR28, a novel radiotracer for imaging the TSPO 18 kDa with PET |
007608 |
Aaron Reynolds [Australie] ; Raphy Hanani [Australie] ; David Hibbs [Australie] ; Annelaure Damont [France] ; Eleonora Da Pozzo [Italie] ; Silvia Selleri [Italie] ; Frédéric Dolle [France] ; Claudia Martini [Italie] ; Michael Kassiou [Australie] | Pyrazolo[1,5-a]pyrimidine acetamides: 4-Phenyl alkyl ether derivatives as potent ligands for the 18 kDa translocator protein (TSPO) |
007870 |
Abraham Martin [France] ; Raphaël Boisgard [France] ; Benoit Theze [France] ; Nadja Van Camp [France] ; Bertrand Kuhnast [France] ; Annelaure Damont [France] ; Michael Kassiou [Australie] ; Frédéric Dolle [France] ; Bertrand Tavitian [France] | Evaluation of the PBR/TSPO radioligand [18F]DPA-714 in a rat model of focal cerebral ischemia |
008134 |
Frédéric Dolle [France] ; Christopher Luus [Australie] ; Aaron Reynolds [Australie] ; Michael Kassiou [Australie] | Radiolabelled Molecules for Imaging the Translocator Protein (18 kDa) Using Positron Emission Tomography |
008752 |
Annelaure Damont [France] ; Françoise Hinnen [France] ; Bertrand Kuhnast [France] ; Marie-Anne Schöllhorn-Peyronneau [France] ; Michelle James [Australie] ; Christopher Luus [Australie] ; Bertrand Tavitian [France] ; Michael Kassiou [Australie] ; Frédéric Dollé [France] | Radiosynthesis of [18F]DPA‐714, a selective radioligand for imaging the translocator protein (18 kDa) with PET |
008843 |
Laurent Besret [France] ; Frédéric Dollé [France] ; Anne-Sophie Hérard [France] ; Martine Guillermier [France] ; Stéphane Demphel [France] ; Françoise Hinnen [France] ; Christine Coulon [France] ; Michèle Ottaviani [France] ; Michel Bottlaender [France] ; Philippe Hantraye [France] ; Michael Kassiou [Australie] | Dopamine D1 receptor imaging in the rodent and primate brain using the isoquinoline (+)‐[11C]A‐69024 and positron emission tomography |
009168 |
Nicolas Giboureau [France, Australie] ; Patrick Emond [France] ; Roger R. Fulton [Australie] ; David J. Henderson [Australie] ; Sylvie Chalon [France] ; Lucette Garreau [France] ; Peter Roselt [Australie] ; Stefan Eberl [Australie] ; Sylvie Mavel [France] ; Sylvie Bodard [France] ; Michael J. Fulham [Australie] ; Denis Guilloteau [France] ; Michael Kassiou [Australie] | Ex vivo and in vivo evaluation of (2R,3R)‐5‐[18F]‐fluoroethoxy‐ and fluoropropoxy‐benzovesamicol, as PET radioligands for the vesicular acetylcholine transporter |
009212 |
Alan Kozikowski [États-Unis] ; Sheela Chellappan [États-Unis] ; David Henderson [Australie] ; Roger Fulton [Australie] ; Nicolas Giboureau [France] ; Yingxian Xiao [États-Unis] ; Zhi-Liang Wei [États-Unis] ; Denis Guilloteau [France] ; Patrick Emond [France] ; Frederic Dolle [France] ; Kenneth Kellar [États-Unis] ; Michael Kassiou [Australie] | Acetylenic Pyridines for Use in PET Imaging of Nicotinic Receptors |
009649 |
Mitchell Quinlivan [France, Australie] ; Sylvie Chalon [France] ; Jackie Vergote [France] ; Jasmine Henderson [Australie] ; Andrew Katsifis [Australie] ; Michael Kassiou [Australie] ; Denis Guilloteau [France] | Decreased vesicular acetylcholine transporter and α4β2 nicotinic receptor density in the rat brain following 192 IgG-saporin immunolesioning |
009B84 |
Johnny Vercouillie [France] ; Sylvie Mavel [France] ; Laurent Galineau [France] ; Tiziana Ragusa [France] ; Robert Innis [États-Unis] ; Michael Kassiou [Australie] ; Sylvie Chalon [France] ; Frédéric Dolle [France] ; Jean-Claude Besnard [France] ; Denis Guilloteau [France] ; Patrick Emond [France] | Synthesis and in vitro evaluation of novel derivatives of diphenylsulfide as serotonin transporter ligands |
009B85 |
Thaer Assaad [France] ; Sylvie Mavel [France] ; Stanley M. Parsons [États-Unis] ; Shane Kruse [États-Unis] ; Laurent Galineau [France] ; Hassan Allouchi [France] ; Michael Kassiou [Australie] ; Sylvie Chalon [France] ; Denis Guilloteau [France] ; Patrick Emond [France] | Synthesis and in vitro evaluation of N-substituted aza-trozamicol analogs as vesicular acetylcholine transporter ligands |
00A417 |
Michelle L. James [Australie] ; Roger R. Fulton [Australie] ; David J. Henderson [Australie] ; Stefan Eberl [Australie] ; Steven R. Meikle [Australie] ; Sally Thomson [Australie] ; Robin D. Allan [Australie] ; Frederic Dolle [France] ; Michael J. Fulham [Australie] ; Michael Kassiou [Australie] | Synthesis and in vivo evaluation of a novel peripheral benzodiazepine receptor PET radioligand |
00A418 |
Yolanda Zea-Ponce [France] ; Sylvie Mavel [France] ; Thaer Assaad [France] ; Shane E. Kruse [États-Unis] ; Stanley M. Parsons [États-Unis] ; Patrick Emond [France] ; Sylvie Chalon [France] ; Nicolas Giboureau [France, Australie] ; Michael Kassiou [Australie] ; Denis Guilloteau [France] | Synthesis and in vitro evaluation of new benzovesamicol analogues as potential imaging probes for the vesicular acetylcholine transporter |
00A881 |
Frédéric Dollé [France] ; Héric Valette [France] ; Stéphane Demphel [France] ; Christine Coulon [France] ; Michelle Ottaviani [France] ; Michel Bottlaender [France] ; Michael Kassiou [Australie] | Radiosynthesis and in vivo evaluation of [11C]Ro‐647312: a novel NR1/2B subtype selective NMDA receptor radioligand |
00B026 |
Gaëlle Roger [France] ; Béatrice Lagnel [France] ; Laurent Besret [France] ; Yann Bramoulle [France] ; Christine Coulon [France] ; Michelle Ottaviani [France] ; Michael Kassiou [Australie] ; Michel Bottlaender [France] ; Heric Valette [France] ; Frédéric Dolle [France] | Synthesis, radiosynthesis and in vivo evaluation of 5-[3-(4-benzylpiperidin-1-yl)prop-1-ynyl]-1,3-dihydrobenzoimidazol-2-[11C]one, as a potent NR1A/2B subtype selective NMDA PET radiotracer |
00B027 |
Mitchell Quinlivan [Australie] ; Filomena Mattner [Australie] ; Vahan Papazian [Australie] ; JIA ZHOU [États-Unis] ; Andrew Katsifis [Australie] ; Patrick Emond [France] ; Sylvie Chalon [France] ; Alan Kozikowski [États-Unis] ; Denis Guilloteau [France] ; Michael Kassiou [Australie] | Synthesis and evaluation of iodine-123 labelled tricyclic tropanes as radioligands for the serotonin transporter |
00B090 |
Andrew Ratsifis [Australie] ; Karine Mardon [Australie] ; Filomena Mattner [Australie] ; Christian Loc'H [France] ; Meredith E. Mcphee [Australie] ; Branko Dikic [Australie] ; Michael Kassiou [Australie] ; Damon D. Ridley [Australie] | Pharmacological evaluation of (S)-8-[123I]iodobretazenil: a radioligand for in vivo studies of central benzodiazepine receptors |
00BF46 |
Michael Kassiou [Australie] ; Christian Loc'H [France] ; Andrew Katsifis [Australie] ; Vahan Papazian [Australie] ; Filomena Mattner [Australie] ; Branko Dikic [Australie] ; Bernard Mazière [France] | Radiosynthesis of bromine‐76 and iodine‐123 labelled enantiomers of A‐69024: radioligands for dopamine D1 receptor studies using PET and SPECT |
00D150 |
Michael Kassiou [Australie] ; Karine Mardon [Australie] ; Andrew G. Katsifis [Australie] ; Ljubco Najdovski [Australie] ; Branko Dikic [Australie] ; Filomena Mattner [Australie] ; Richard M. Lambrecht [France] ; Rodney J. Hicks [Australie] ; Peter Eu [Australie] ; Christian Loc'H [France] | Radiosynthesis of [123I]N-methyl-4-iododexetimide and [123I]N-methyl-4-iodolevetimide: In vitro and in vivo characterisation of binding to muscarinic receptors in the rat heart |
00D482 |
Michael Kassiou [Australie, France] ; Christian Loc'H [France] ; Veronique Strijckmans [France] ; Andrew Katsifis [Australie] ; Richard M. Lambrecht [Australie] ; Mariannick Maziere [France] ; Bernard Maziere [France] | Synthesis of [76Br]4‐bromodexetimide and [76Br]4‐bromolevetimide: Radiotracers for studying muscarinic cholinergic receptors using PET |